MolecularFormula: | C20H21FN6O | Melting Point: | |
---|---|---|---|
Molecular Weight: | 380.42 | Packaging: | |
Appearance: | ProductionCapacity: | Kgs~Tons | |
Purity: | 99%+ | Productuse: |
Selitrectinib (LOXO-195) is a next-generation TRK kinaseinhibitor (TKI), with IC50sof 0.6 nM, <2.5 nM for TRKA and TRKC respectively.